PI3K-Akt signaling pathway;MAPK signaling pathway;apoptosis(凋亡);DNA damage( DNA 损伤);RTK(受体酪氨酸激酶)
货号 |
靶点 |
产品名称 |
国内报价(元) |
K1001 |
JNK |
SP600125 |
2mg:700,5mg:1000,10mg:1500 |
K1002 |
HIF |
2-Methoxyestradiol |
2mg:700,5mg:1000,10mg:1500 |
K1003 |
VEGFR |
Linifanib (ABT-869) |
2mg:1100,5mg:1500,10mg:2100 |
K1004 |
PARP |
ABT-888 (Veliparib) |
2mg:900,5mg:1200,10mg:1700 |
K1005 |
PARP |
Olaparib(AZD2281) |
2mg:700,5mg:1000,10mg:1500 |
K1006 |
Bcr-Abl |
Imatinib Mesylate |
2mg:500,5mg:800,10mg:1100 |
K1007 |
PDGFR |
Imatinib (Gleevec) |
2mg:500,5mg:800,10mg:1100 |
K1008 |
VEGFR |
XL-184(Cabozantinib) |
2mg:900,5mg:1200,10mg:1700 |
K1009 |
PARP |
Iniparib (BSI-201) |
2mg:700,5mg:1000,10mg:1500 |
K1010 |
Flt |
AC220 (Quizartinib) |
2mg:1500,5mg:2100,10mg:3000 |
K1011 |
TNF-alpha |
Pomalidomide |
2mg:700,5mg:1000,10mg:1500 |
K1012 |
Aurora Kinase |
ENMD-2076 |
2mg:1300,5mg:1900,10mg:2800 |
K1013 |
HDAC |
Entinostat (MS-275, SNDX-275) |
2mg:700,5mg:1000,10mg:1500 |
K1014 |
MEK |
U0126-EtOH |
2mg:500,5mg:800,10mg:1100 |
K1015 |
Bcl-2 |
Obatoclax mesylate (GX15-070) |
2mg:1100,5mg:1500,10mg:2100 |
K1016 |
Antimetabolites |
Cisplatin |
2mg:500,5mg:800,10mg:1100 |
K1017 |
EGFR |
Erlotinib hydrochloride |
2mg:500,5mg:800,10mg:1100 |
K1018 |
EGFR |
Gefitinib (Iressa) |
2mg:500,5mg:800,10mg:1100 |
K1019 |
aromatase (CYP19) |
Exemestane |
2mg:500,5mg:800,10mg:1100 |
K1020 |
Proteasome |
Bortezomib (Velcade) |
2mg:700,5mg:1000,10mg:1500 |